PDB Information

PDB3TZA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: synthesis, resolution, pharmacology, and crystal structure
Szymanska, E., Frydenvang, K., Contreras-Sanz, A., Pickering, D.S., Frola, E., Serafimoska, Z., Nielsen, B., Kastrup, J.S., Johansen, T.N.
J.Med.Chem.
HeaderMembrane Protein
Released2011-09-27
Resolution1.900
CATH Insert Date30 Oct, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped
B 29 Nov, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3tzaA01 01 Dec, 2011 3.40.190.10 Assigned
3tzaA02 01 Dec, 2011 3.40.190.10 Assigned
3tzaB01 01 Dec, 2011 3.40.190.10 Assigned
3tzaB02 01 Dec, 2011 3.40.190.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2