PDB Information

PDB3TKH
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Pyridyl aminothiazoles as potent inhibitors of Chk1 with slow dissociation rates.
Dudkin, V.Y., Rickert, K., Kreatsoulas, C., Wang, C., Arrington, K.L., Fraley, M.E., Hartman, G.D., Yan, Y., Ikuta, M., Stirdivant, S.M., Drakas, R.A., Walsh, E.S., Hamilton, K., Buser, C.A., Lobell, R.B., Sepp-Lorenzino, L.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-08-26
Resolution1.790
CATH Insert Date27 May, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 May, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3tkhA01 08 Jun, 2012 3.30.200.20 Assigned
3tkhA02 08 Jun, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14757 CHK1_HUMAN Homo sapiens Serine/threonine-protein kinase Chk1