PDB 3sx0
PDB Information
| PDB | 3SX0 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Bromo-deaza-SAH: a potent and selective DOT1L inhibitor.
Bioorg. Med. Chem.
|
| Header | Transferase |
| Released | 2011-07-14 |
| Resolution | 2.280 |
| CATH Insert Date | 07 Aug, 2011 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Aug, 2011 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3sx0A01 | 12 Aug, 2011 | 1.10.260.60 | Assigned |
| 3sx0A02 | 12 Aug, 2011 | 3.40.50.150 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q8TEK3 | DOT1L_HUMAN | Homo sapiens | Histone-lysine N-methyltransferase, H3 lysine-79 specific |
