PDB 3she
PDB Information
| PDB | 3SHE |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2011-06-16 |
| Resolution | 2.250 |
| CATH Insert Date | 08 Jan, 2012 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 09 Jan, 2012 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3sheA01 | 16 Jan, 2012 | 3.30.200.20 | Assigned |
| 3sheA02 | 16 Jan, 2012 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q16644 | MAPK3_HUMAN | Homo sapiens | MAP kinase-activated protein kinase 3 |
