PDB 3sc1
PDB Information
| PDB | 3SC1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Novel isoquinolone PDK1 inhibitors discovered through fragment-based lead discovery.
J Comput Aided Mol Des
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2011-06-06 |
| Resolution | 2.700 |
| CATH Insert Date | 30 Oct, 2011 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Nov, 2011 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3sc1A01 | 01 Dec, 2011 | 3.30.200.20 | Assigned |
| 3sc1A02 | 01 Dec, 2011 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O15530 | PDPK1_HUMAN | Homo sapiens | 3-phosphoinositide-dependent protein kinase 1 |
