PDB Information

PDB3RZ3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
An allosteric inhibitor of the human cdc34 ubiquitin conjugating enzyme
Ceccarelli, D.F., Tang, X., Pelletier, B., Orlicky, S., Xie, W., Plantevin, V., Neculai, D., Chou, Y.C., Ogunjimi, A., Al-Hakim, A., Varelas, X., Koszela, J., Wasney, G.A., Vedadi, M., Dhe-Paganon, S., Cox, S., Xu, S., Lopez-Girona, A., Mercurio, F., Wrana, J., Durocher, D., Meloche, S., Webb, D.R., Tyers, M., Sicheri, F.
Cell(Cambridge,Mass.)
HeaderLigase/Ligase Inhibitor
Released2011-05-11
Resolution2.300
CATH Insert Date24 Jul, 2011

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 25 Jul, 2011 Chopped
B 25 Jul, 2011 Chopped
C 25 Jul, 2011 Chopped
D 25 Jul, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3rz3A00 04 Aug, 2011 3.10.110.10 Assigned
3rz3B00 04 Aug, 2011 3.10.110.10 Assigned
3rz3C00 04 Aug, 2011 3.10.110.10 Assigned
3rz3D00 04 Aug, 2011 3.10.110.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P49427 UB2R1_HUMAN Homo sapiens Ubiquitin-conjugating enzyme E2 R1
P49427 UB2R1_HUMAN Homo sapiens Ubiquitin-conjugating enzyme E2 R1
P49427 UB2R1_HUMAN Homo sapiens Ubiquitin-conjugating enzyme E2 R1
P49427 UB2R1_HUMAN Homo sapiens Ubiquitin-conjugating enzyme E2 R1