PDB 3rwp

PDB Information

PDB3RWP
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of Novel, Potent, and Selective Inhibitors of 3-Phosphoinositide-Dependent Kinase (PDK1).
Murphy, S.T., Alton, G., Bailey, S., Baxi, S.M., Burke, B.J., Chappie, T.A., Ermolieff, J., Ferre, R., Greasley, S., Hickey, M., Humphrey, J., Kablaoui, N., Kath, J., Kazmirski, S., Kraus, M., Kupchinsky, S., Li, J., Lingardo, L., Marx, M.A., Richter, D., Tanis, S.P., Tran, K., Vernier, W., Xie, Z., Yin, M.J., Yu, X.H.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2011-05-09
Resolution1.920
CATH Insert Date20 Nov, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3rwpA01 01 Dec, 2011 3.30.200.20 Assigned
3rwpA02 01 Dec, 2011 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1