PDB Information

PDB3ROC
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Substituted N-aryl-6-pyrimidinones: A new class of potent, selective, and orally active p38 MAP kinase inhibitors.
Devadas, B., Selness, S.R., Xing, L., Madsen, H.M., Marrufo, L.D., Shieh, H., Messing, D.M., Yang, J.Z., Morgan, H.M., Anderson, G.D., Webb, E.G., Zhang, J., Devraj, R.V., Monahan, J.B.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-04-25
Resolution1.700
CATH Insert Date19 Jun, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Jun, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3rocA01 22 Jun, 2011 3.30.200.20 Assigned
3rocA02 22 Jun, 2011 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q16539 MK14_HUMAN Homo sapiens Mitogen-activated protein kinase 14