PDB 3ro4
PDB Information
| PDB | 3RO4 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Optimization of a pyrazole hit from FBDD into a novel series of indazoles as ketohexokinase inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2011-04-25 |
| Resolution | 2.600 |
| CATH Insert Date | 07 Aug, 2011 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Aug, 2011 | Chopped |
| B | 08 Aug, 2011 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3ro4A00 | 01 Feb, 2013 | 3.40.1190.20 | Assigned |
| 3ro4B00 | 08 Feb, 2013 | 3.40.1190.20 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P50053 | KHK_HUMAN | Homo sapiens | Ketohexokinase |
| P50053 | KHK_HUMAN | Homo sapiens | Ketohexokinase |
