PDB Information

PDB3R8A
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a Series of Imidazo[4,5-b]pyridines with Dual Activity at Angiotensin II Type 1 Receptor and Peroxisome Proliferator-Activated Receptor-gamma.
Casimiro-Garcia, A., Filzen, G.F., Flynn, D., Bigge, C.F., Chen, J., Davis, J.A., Dudley, D.A., Edmunds, J.J., Esmaeil, N., Geyer, A., Heemstra, R.J., Jalaie, M., Ohren, J.F., Ostroski, R., Ellis, T., Schaum, R.P., Stoner, C.
J.Med.Chem.
HeaderNuclear Protein
Released2011-03-23
Resolution2.410
CATH Insert Date27 May, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 May, 2012 Chopped
B 28 May, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3r8aA00 08 Jun, 2012 1.10.565.10 Assigned
3r8aB00 08 Jun, 2012 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma