PDB Information

PDB3QKD
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Quinazoline sulfonamides as dual binders of the proteins B-cell lymphoma 2 and B-cell lymphoma extra long with potent proapoptotic cell-based activity.
Sleebs, B.E., Czabotar, P.E., Fairbrother, W.J., Fairlie, W.D., Flygare, J.A., Huang, D.C., Kersten, W.J., Koehler, M.F., Lessene, G., Lowes, K., Parisot, J.P., Smith, B.J., Smith, M.L., Souers, A.J., Street, I.P., Yang, H., Baell, J.B.
J.Med.Chem.
HeaderApoptosis/Inhibitor
Released2011-01-31
Resolution2.020
CATH Insert Date10 Apr, 2011

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2011 Chopped
B 11 Apr, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3qkdA00 13 Apr, 2011 Holding pen
3qkdB00 12 Apr, 2011 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1