PDB Information

PDB3Q4C
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
The crystal structure of BRAF in complex with an organoruthenium inhibitor reveals a mechanism for inhibition of an active form of BRAF kinase.
Xie, P., Streu, C., Qin, J., Bregman, H., Pagano, N., Meggers, E., Marmorstein, R.
Biochemistry
HeaderTransferase/Transferase Inhibitor
Released2010-12-23
Resolution3.200
CATH Insert Date06 Mar, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Mar, 2011 Chopped
B 06 Mar, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3q4cA01 10 Mar, 2011 3.30.200.20 Assigned
3q4cA02 10 Mar, 2011 1.10.510.10 Assigned
3q4cB01 10 Mar, 2011 3.30.200.20 Assigned
3q4cB02 10 Mar, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf