PDB Information

PDB3Q3T
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Biphenyl/diphenyl ether renin inhibitors: Filling the S1 pocket of renin via the S3 pocket.
Yuan, J., Simpson, R.D., Zhao, W., Tice, C.M., Xu, Z., Cacatian, S., Jia, L., Flaherty, P.T., Guo, J., Ishchenko, A., Wu, Z., McKeever, B.M., Scott, B.B., Bukhtiyarov, Y., Berbaum, J., Panemangalore, R., Bentley, R., Doe, C.P., Harrison, R.K., McGeehan, G.M., Singh, S.B., Dillard, L.W., Baldwin, J.J., Claremon, D.A.
Bioorg.Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2010-12-22
Resolution2.600
CATH Insert Date07 Aug, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Aug, 2011 Chopped
B 08 Aug, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3q3tA01 04 Nov, 2013 2.40.70.10 Assigned
3q3tA02 04 Nov, 2013 2.40.70.10 Assigned
3q3tB01 04 Nov, 2013 2.40.70.10 Assigned
3q3tB02 04 Nov, 2013 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00797 RENI_HUMAN Homo sapiens Renin
P00797 RENI_HUMAN Homo sapiens Renin
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