PDB Information

PDB3Q0T
MethodX-RAY DIFFRACTION
Host OrganismPichia pastoris
Gene SourceHomo sapiens
Primary Citation
Discovery of 7-oxo-pyrrolopyridines as potent and selective inhibitors of dpp4
Wang, W., Devasthale, P., Wang, A., Egan, D., Morgan, N., Cap, M., Fura, A., Klei, H.E., Kish, K., Sun, L., Levesque, P., Zahler, R., Kirby, M., Hamann, L.G.
To be Published
HeaderHydrolase/Hydrolase Inhibitor
Released2010-12-16
Resolution2.400
CATH Insert Date27 May, 2012

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 May, 2012 Chopped
B 28 May, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3q0tA01 08 Jun, 2012 3.40.50.1820 Assigned
3q0tA02 08 Jun, 2012 2.140.10.30 Assigned
3q0tB01 08 Jun, 2012 3.40.50.1820 Assigned
3q0tB02 08 Jun, 2012 2.140.10.30 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4