PDB Information

PDB3PYY
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of a Cell-Permeable, Small-Molecule c-Abl Kinase Activator that Binds to the Myristoyl Binding Site.
Yang, J., Campobasso, N., Biju, M.P., Fisher, K., Pan, X.Q., Cottom, J., Galbraith, S., Ho, T., Zhang, H., Hong, X., Ward, P., Hofmann, G., Siegfried, B., Zappacosta, F., Washio, Y., Cao, P., Qu, J., Bertrand, S., Wang, D.Y., Head, M.S., Li, H., Moores, S., Lai, Z., Johanson, K., Burton, G., Erickson-Miller, C., Simpson, G., Tummino, P., Copeland, R.A., Oliff, A.
Chem.Biol.
HeaderTransferase
Released2010-12-13
Resolution1.850
CATH Insert Date13 Mar, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 13 Mar, 2011 Chopped
B 13 Mar, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3pyyA01 18 Mar, 2011 3.30.200.20 Assigned
3pyyA02 18 Mar, 2011 1.10.510.10 Assigned
3pyyB01 18 Mar, 2011 3.30.200.20 Assigned
3pyyB02 18 Mar, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1