PDB Information

PDB3PSD
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Non-oxime pyrazole based inhibitors of B-Raf kinase.
Newhouse, B.J., Hansen, J.D., Grina, J., Welch, M., Topalov, G., Littman, N., Callejo, M., Martinson, M., Galbraith, S., Laird, E.R., Brandhuber, B.J., Vigers, G., Morales, T., Woessner, R., Randolph, N., Lyssikatos, J., Olivero, A.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2010-12-01
Resolution3.600
CATH Insert Date22 May, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 May, 2011 Chopped
B 23 May, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3psdA01 26 May, 2011 3.30.200.20 Assigned
3psdA02 26 May, 2011 1.10.510.10 Assigned
3psdB01 26 May, 2011 3.30.200.20 Assigned
3psdB02 26 May, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf