PDB Information

PDB3PPK
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Non-oxime inhibitors of B-Raf(V600E) kinase.
Ren, L., Wenglowsky, S., Miknis, G., Rast, B., Buckmelter, A.J., Ely, R.J., Schlachter, S., Laird, E.R., Randolph, N., Callejo, M., Martinson, M., Galbraith, S., Brandhuber, B.J., Vigers, G., Morales, T., Voegtli, W.C., Lyssikatos, J.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2010-11-24
Resolution3.000
CATH Insert Date06 Feb, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Feb, 2011 Chopped
B 07 Feb, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3ppkA01 19 Feb, 2011 3.30.200.20 Assigned
3ppkA02 19 Feb, 2011 1.10.510.10 Assigned
3ppkB01 19 Feb, 2011 3.30.200.20 Assigned
3ppkB02 19 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf