PDB 3p9j
PDB Information
| PDB | 3P9J |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2010-10-17 |
| Resolution | 2.800 |
| CATH Insert Date | 27 Mar, 2011 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 28 Mar, 2011 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3p9jA01 | 01 Apr, 2011 | 3.30.200.20 | Assigned |
| 3p9jA02 | 01 Apr, 2011 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O14965 | AURKA_HUMAN | Homo sapiens | Aurora kinase A |
