PDB 3oq1
PDB Information
| PDB | 3OQ1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | The synthesis and SAR of novel diarylsulfone 11beta-HSD1 inhibitors
Bioorg.Med.Chem.Lett.
|
| Header | Oxidoreductase/Oxidoreductase Inhibitor |
| Released | 2010-09-02 |
| Resolution | 2.600 |
| CATH Insert Date | 24 Jul, 2011 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 25 Jul, 2011 | Chopped |
| B | 25 Jul, 2011 | Chopped |
| C | 25 Jul, 2011 | Chopped |
| D | 25 Jul, 2011 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3oq1A00 | 04 Aug, 2011 | 3.40.50.720 | Assigned |
| 3oq1B00 | 04 Aug, 2011 | 3.40.50.720 | Assigned |
| 3oq1C00 | 04 Aug, 2011 | 3.40.50.720 | Assigned |
| 3oq1D00 | 04 Aug, 2011 | 3.40.50.720 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
| P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
