PDB 3o9v
PDB Information
| PDB | 3O9V |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of a 3-Pyridylacetic Acid Derivative (TAK-100) as a Potent, Selective and Orally Active Dipeptidyl Peptidase IV (DPP-4) Inhibitor.
J.Med.Chem.
|
| Header | Hydrolase,Signaling Protein/Inhibitor |
| Released | 2010-08-04 |
| Resolution | 2.750 |
| CATH Insert Date | 13 Feb, 2011 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Feb, 2011 | Chopped |
| B | 14 Feb, 2011 | Chopped |
| C | 14 Feb, 2011 | Chopped |
| D | 14 Feb, 2011 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3o9vA01 | 18 Feb, 2011 | 2.140.10.30 | Assigned |
| 3o9vA02 | 18 Feb, 2011 | 3.40.50.1820 | Assigned |
| 3o9vB01 | 18 Feb, 2011 | 2.140.10.30 | Assigned |
| 3o9vB02 | 18 Feb, 2011 | 3.40.50.1820 | Assigned |
| 3o9vC01 | 18 Feb, 2011 | 2.140.10.30 | Assigned |
| 3o9vC02 | 18 Feb, 2011 | 3.40.50.1820 | Assigned |
| 3o9vD01 | 18 Feb, 2011 | 2.140.10.30 | Assigned |
| 3o9vD02 | 18 Feb, 2011 | 3.40.50.1820 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 |
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 |
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 |
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 |
