PDB Information

PDB3NPC
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
X-ray crystal structure of JNK2 complexed with the p38alpha inhibitor BIRB796: Insights into the rational design of DFG-out binding MAP kinase inhibitors.
Kuglstatter, A., Ghate, M., Tsing, S., Villasenor, A.G., Shaw, D., Barnett, J.W., Browner, M.F.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2010-06-28
Resolution2.350
CATH Insert Date15 Aug, 2010

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2010 Chopped
B 16 Aug, 2010 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3npcA01 17 Feb, 2011 3.30.200.20 Assigned
3npcA02 17 Feb, 2011 1.10.510.10 Assigned
3npcB01 16 Feb, 2011 3.30.200.20 Assigned
3npcB02 16 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P45984 MK09_HUMAN Homo sapiens Mitogen-activated protein kinase 9
P45984 MK09_HUMAN Homo sapiens Mitogen-activated protein kinase 9