PDB Information

PDB3MO2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Adding a lysine mimic in the design of potent inhibitors of histone lysine methyltransferases.
Chang, Y., Ganesh, T., Horton, J.R., Spannhoff, A., Liu, J., Sun, A., Zhang, X., Bedford, M.T., Shinkai, Y., Snyder, J.P., Cheng, X.
J.Mol.Biol.
HeaderTransferase
Released2010-04-22
Resolution2.490
CATH Insert Date04 Jul, 2010

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 04 Jul, 2010 Chopped
B 04 Jul, 2010 Chopped
C 04 Jul, 2010 Chopped
D 04 Jul, 2010 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3mo2A00 19 Aug, 2010 2.170.270.10 Assigned
3mo2B00 19 Aug, 2010 2.170.270.10 Assigned
3mo2C00 19 Aug, 2010 2.170.270.10 Assigned
3mo2D00 19 Aug, 2010 2.170.270.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1