PDB Information

PDB3MBL
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based design and synthesis of pyrrole derivatives as MEK inhibitors.
Wallace, M.B., Adams, M.E., Kanouni, T., Mol, C.D., Dougan, D.R., Feher, V.A., O'Connell, S.M., Shi, L., Halkowycz, P., Dong, Q.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2010-03-25
Resolution2.600
CATH Insert Date15 Aug, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3mblA01 20 Sep, 2013 3.30.200.20 Assigned
3mblA02 20 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q02750 MP2K1_HUMAN Homo sapiens Dual specificity mitogen-activated protein kinase kinase 1