PDB 3lzb
PDB Information
| PDB | 3LZB |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Imidazo[2,1-b]thiazoles: multitargeted inhibitors of both the insulin-like growth factor receptor and members of the epidermal growth factor family of receptor tyrosine kinases.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2010-03-01 |
| Resolution | 2.700 |
| CATH Insert Date | 06 Mar, 2011 |
PDB Images (17)
PDB Prints
PDB Chains (8)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 06 Mar, 2011 | Chopped |
| B | 06 Mar, 2011 | Chopped |
| C | 06 Mar, 2011 | Chopped |
| D | 06 Mar, 2011 | Chopped |
| E | 06 Mar, 2011 | Rejected |
| F | 06 Mar, 2011 | Rejected |
| G | 06 Mar, 2011 | Rejected |
| H | 06 Mar, 2011 | Rejected |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3lzbA01 | 10 Mar, 2011 | 3.30.200.20 | Assigned |
| 3lzbA02 | 10 Mar, 2011 | 1.10.510.10 | Assigned |
| 3lzbB01 | 10 Mar, 2011 | 3.30.200.20 | Assigned |
| 3lzbB02 | 10 Mar, 2011 | 1.10.510.10 | Assigned |
| 3lzbC01 | 10 Mar, 2011 | 3.30.200.20 | Assigned |
| 3lzbC02 | 10 Mar, 2011 | 1.10.510.10 | Assigned |
| 3lzbD01 | 09 Mar, 2011 | 3.30.200.20 | Assigned |
| 3lzbD02 | 09 Mar, 2011 | 1.10.510.10 | Assigned |
UniProtKB Entries (8)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
| P00533 | EGFR_HUMAN | Homo sapiens | Epidermal growth factor receptor |
