PDB Information

PDB3LXG
MethodX-RAY DIFFRACTION
Host Organismbaculovirus
Gene SourceRattus norvegicus
Primary Citation
Discovery of imidazo[1,5-a]pyrido[3,2-e]pyrazines as a new class of phosphodiesterase 10A inhibitiors.
Hofgen, N., Stange, H., Schindler, R., Lankau, H.J., Grunwald, C., Langen, B., Egerland, U., Tremmel, P., Pangalos, M.N., Marquis, K.L., Hage, T., Harrison, B.L., Malamas, M.S., Brandon, N.J., Kronbach, T.
J.Med.Chem.
HeaderHydrolase
Released2010-02-25
Resolution2.300
CATH Insert Date23 May, 2010

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 24 May, 2010 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3lxgA00 08 Feb, 2013 1.10.1300.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9QYJ6 PDE10_RAT Rattus norvegicus cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A