PDB Information

PDB3L9M
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Azole-based inhibitors of AKT/PKB for the treatment of cancer.
Zeng, Q., Allen, J.G., Bourbeau, M.P., Wang, X., Yao, G., Tadesse, S., Rider, J.T., Yuan, C.C., Hong, F.T., Lee, M.R., Zhang, S., Lofgren, J.A., Freeman, D.J., Yang, S., Li, C., Tominey, E., Huang, X., Hoffman, D., Yamane, H.K., Fotsch, C., Dominguez, C., Hungate, R., Zhang, X.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2010-01-05
Resolution1.900
CATH Insert Date23 Jan, 2011

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped
B 24 Jan, 2011 Chopped
C 24 Jan, 2011 Rejected
D 24 Jan, 2011 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3l9mA01 17 Feb, 2011 1.10.510.10 Assigned
3l9mA02 17 Feb, 2011 3.30.200.20 Assigned
3l9mB01 17 Feb, 2011 1.10.510.10 Assigned
3l9mB02 17 Feb, 2011 3.30.200.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P17612 KAPCA_HUMAN Homo sapiens cAMP-dependent protein kinase catalytic subunit alpha
P17612 KAPCA_HUMAN Homo sapiens cAMP-dependent protein kinase catalytic subunit alpha