PDB Information

PDB3L8X
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Pyrazolo-Pyrimidines: A Novel Heterocyclic Scaffold for Potent and Selective P38 Alpha Inhibitors.
Das, J., Moquin, R.V., Pitt, S., Zhang, R., Shen, D.R., Mcintyre, K.W., Gillooly, K., Doweyko, A.M., Sack, J.S., Zhang, H., Kiefer, S.E., Kish, K., Mckinnon, M., Barrish, J.C., Dodd, J.H., Schieven, G.L., Leftheris, K.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2010-01-04
Resolution2.400
CATH Insert Date04 Mar, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3l8xA01 06 Jul, 2010 3.30.200.20 Assigned
3l8xA02 06 Jul, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q16539 MK14_HUMAN Homo sapiens Mitogen-activated protein kinase 14