PDB Information

PDB3L8V
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHomo sapiens
Primary Citation
Design, synthesis and structure-activity relationships of novel biarylamine-based Met kinase inhibitors.
Williams, D.K., Chen, X.T., Tarby, C., Kaltenbach, R., Cai, Z.W., Tokarski, J.S., An, Y., Sack, J.S., Wautlet, B., Gullo-Brown, J., Henley, B.J., Jeyaseelan, R., Kellar, K., Manne, V., Trainor, G.L., Lombardo, L.J., Fargnoli, J., Borzilleri, R.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2010-01-04
Resolution2.400
CATH Insert Date09 May, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 May, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3l8vA01 06 Jul, 2010 3.30.200.20 Assigned
3l8vA02 06 Jul, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor