PDB Information

PDB3KXO
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of an oral potent selective inhibitor of hematopoietic prostaglandin D synthase
Carron, C.P., Trujillo, J.I., Olson, K.L., Huang, W., Hamper, B.C., Dice, T., Neal, B.E., Pelc, M.J., Day, J., Rohrer, D.C., Kiefer, J.R., Moon, J.B., Schweitzer, B.A., Blake, T.D., Turner, S.R., Woerndle, R., Case, B.L., Bono, C.P., Dilworth, V.M., Funckes-Shippy, C.L., Hood, B.L., Jerome, G.M., Kornmeier, C.M., Radabaugh, M.R., Williams, M.L., Davies, M.S., Wegner, C.D., Welsch, D.J., Abraham, W.M., Warren, C.J., Dowty, M.E., Hua, F., Zutshi, A., Yang, J.Z., Thorarensen, A.
TO BE PUBLISHED
HeaderIsomerase
Released2009-12-03
Resolution2.100
CATH Insert Date05 Sep, 2010

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Sep, 2010 Chopped
B 06 Sep, 2010 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3kxoA01 26 Sep, 2010 3.40.30.10 Assigned
3kxoA02 26 Sep, 2010 1.20.1050.10 Assigned
3kxoB01 27 Sep, 2010 3.40.30.10 Assigned
3kxoB02 27 Sep, 2010 1.20.1050.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60760 HPGDS_HUMAN Homo sapiens Hematopoietic prostaglandin D synthase
O60760 HPGDS_HUMAN Homo sapiens Hematopoietic prostaglandin D synthase