PDB Information

PDB3KQS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors.
Drinkwater, N., Vu, H., Lovell, K.M., Criscione, K.R., Collins, B.M., Prisinzano, T.E., Poulsen, S.A., McLeish, M.J., Grunewald, G.L., Martin, J.L.
Biochem.J.
HeaderTransferase
Released2009-11-17
Resolution2.010
CATH Insert Date03 Oct, 2010

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 04 Oct, 2010 Chopped
B 04 Oct, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3kqsA00 12 Oct, 2010 3.40.50.150 Assigned
3kqsB00 12 Oct, 2010 3.40.50.150 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P11086 PNMT_HUMAN Homo sapiens Phenylethanolamine N-methyltransferase
P11086 PNMT_HUMAN Homo sapiens Phenylethanolamine N-methyltransferase