PDB Information

PDB3KC1
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based drug design of tricyclic 8H-indeno[1,2-d][1,3]thiazoles as potent FBPase inhibitors.
Tsukada, T., Takahashi, M., Takemoto, T., Kanno, O., Yamane, T., Kawamura, S., Nishi, T.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2009-10-20
Resolution2.250
CATH Insert Date07 Feb, 2010

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 Feb, 2010 Chopped
B 08 Feb, 2010 Chopped
C 08 Feb, 2010 Chopped
D 08 Feb, 2010 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3kc1A01 15 Apr, 2010 3.30.540.10 Assigned
3kc1A02 15 Apr, 2010 3.40.190.80 Assigned
3kc1B01 15 Apr, 2010 3.30.540.10 Assigned
3kc1B02 15 Apr, 2010 3.40.190.80 Assigned
3kc1C01 15 Apr, 2010 3.30.540.10 Assigned
3kc1C02 15 Apr, 2010 3.40.190.80 Assigned
3kc1D01 15 Apr, 2010 3.30.540.10 Assigned
3kc1D02 15 Apr, 2010 3.40.190.80 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P09467 F16P1_HUMAN Homo sapiens Fructose-1,6-bisphosphatase 1
P09467 F16P1_HUMAN Homo sapiens Fructose-1,6-bisphosphatase 1
P09467 F16P1_HUMAN Homo sapiens Fructose-1,6-bisphosphatase 1
P09467 F16P1_HUMAN Homo sapiens Fructose-1,6-bisphosphatase 1