PDB Information

PDB3K5V
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Targeting Bcr-Abl by combining allosteric with ATP-binding-site inhibitors.
Zhang, J., Adrian, F.J., Jahnke, W., Cowan-Jacob, S.W., Li, A.G., Iacob, R.E., Sim, T., Powers, J., Dierks, C., Sun, F., Guo, G.R., Ding, Q., Okram, B., Choi, Y., Wojciechowski, A., Deng, X., Liu, G., Fendrich, G., Strauss, A., Vajpai, N., Grzesiek, S., Tuntland, T., Liu, Y., Bursulaya, B., Azam, M., Manley, P.W., Engen, J.R., Daley, G.Q., Warmuth, M., Gray, N.S.
Nature
HeaderTransferase
Released2009-10-08
Resolution1.740
CATH Insert Date21 Jan, 2010

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 22 Jan, 2010 Chopped
B 22 Jan, 2010 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3k5vA01 10 Aug, 2010 3.30.200.20 Assigned
3k5vA02 10 Aug, 2010 1.10.510.10 Assigned
3k5vB01 10 Aug, 2010 3.30.200.20 Assigned
3k5vB02 10 Aug, 2010 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00520 ABL1_MOUSE Mus musculus Tyrosine-protein kinase ABL1
P00520 ABL1_MOUSE Mus musculus Tyrosine-protein kinase ABL1