PDB 3k5k
PDB Information
| PDB | 3K5K |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of a 2,4-diamino-7-aminoalkoxyquinazoline as a potent and selective inhibitor of histone lysine methyltransferase G9a.
J.Med.Chem.
|
| Header | Transferase |
| Released | 2009-10-07 |
| Resolution | 1.700 |
| CATH Insert Date | 15 Nov, 2009 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 Nov, 2009 | Chopped |
| B | 15 Nov, 2009 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3k5kA00 | 19 Aug, 2010 | 2.170.270.10 | Assigned |
| 3k5kB00 | 19 Aug, 2010 | 2.170.270.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q96KQ7 | EHMT2_HUMAN | Homo sapiens | Histone-lysine N-methyltransferase EHMT2 |
| Q96KQ7 | EHMT2_HUMAN | Homo sapiens | Histone-lysine N-methyltransferase EHMT2 |
