PDB Information

PDB3I0R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHIV-1 M:B_HXB2R
Primary Citation
Substituted tetrahydroquinolines as potent allosteric inhibitors of reverse transcriptase and its key mutants.
Su, D.S., Lim, J.J., Tinney, E., Wan, B.L., Young, M.B., Anderson, K.D., Rudd, D., Munshi, V., Bahnck, C., Felock, P.J., Lu, M., Lai, M.T., Touch, S., Moyer, G., Distefano, D.J., Flynn, J.A., Liang, Y., Sanchez, R., Prasad, S., Yan, Y., Perlow-Poehnelt, R., Torrent, M., Miller, M., Vacca, J.P., Williams, T.M., Anthony, N.J.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2009-06-25
Resolution2.980
CATH Insert Date30 Aug, 2009

PDB Images (12)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 30 Aug, 2009 Chopped
B 30 Aug, 2009 Chopped

CATH Domains (9)

Domain ID Date inserted into CATH Superfamily CATH Status
3i0rA01 10 Mar, 2010 3.10.10.10 Assigned
3i0rA02 10 Mar, 2010 3.30.70.270 Assigned
3i0rA03 10 Mar, 2010 3.30.70.270 Assigned
3i0rA04 10 Mar, 2010 3.30.70.270 Assigned
3i0rA05 10 Mar, 2010 3.30.420.10 Assigned
3i0rB01 10 Mar, 2010 3.10.10.10 Assigned
3i0rB02 10 Mar, 2010 3.30.70.270 Assigned
3i0rB03 10 Mar, 2010 3.30.70.270 Assigned
3i0rB04 10 Mar, 2010 3.30.70.270 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein