PDB Information

PDB3HDN
MethodX-RAY DIFFRACTION
Host Organismunidentified BACULOVIRUS
Gene SourceHomo sapiens
Primary Citation
Design and synthesis of orally bioavailable serum and glucocorticoid-regulated kinase 1 (SGK1) inhibitors.
Hammond, M., Washburn, D.G., Hoang, H.T., Manns, S., Frazee, J.S., Nakamura, H., Patterson, J.R., Trizna, W., Wu, C., Azzarano, L.M., Nagilla, R., Nord, M., Trejo, R., Head, M.S., Zhao, B., Smallwood, A.M., Hightower, K., Laping, N.J., Schnackenberg, C.G., Thompson, S.K.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2009-05-07
Resolution3.100
CATH Insert Date16 Aug, 2009

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3hdnA01 11 Feb, 2010 3.30.200.20 Assigned
3hdnA02 11 Feb, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O00141 SGK1_HUMAN Homo sapiens Serine/threonine-protein kinase Sgk1