PDB 3h0z
PDB Information
| PDB | 3H0Z |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | A class of 2,4-bisanilinopyrimidine Aurora A inhibitors with unusually high selectivity against Aurora B.
J.Med.Chem.
|
| Header | Transferase |
| Released | 2009-04-10 |
| Resolution | 2.920 |
| CATH Insert Date | 16 Aug, 2009 |
PDB Images (10)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Aug, 2009 | Chopped |
| B | 16 Aug, 2009 | Chopped |
| C | 16 Aug, 2009 | Chopped |
CATH Domains (6)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3h0zA01 | 23 Jan, 2010 | 3.30.200.20 | Assigned |
| 3h0zA02 | 23 Jan, 2010 | 1.10.510.10 | Assigned |
| 3h0zB01 | 23 Jan, 2010 | 3.30.200.20 | Assigned |
| 3h0zB02 | 23 Jan, 2010 | 1.10.510.10 | Assigned |
| 3h0zC01 | 23 Jan, 2010 | 3.30.200.20 | Assigned |
| 3h0zC02 | 23 Jan, 2010 | 1.10.510.10 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O14965 | AURKA_HUMAN | Homo sapiens | Aurora kinase A |
| O14965 | AURKA_HUMAN | Homo sapiens | Aurora kinase A |
| O14965 | AURKA_HUMAN | Homo sapiens | Aurora kinase A |
