PDB Information

PDB3GJW
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Synthesis and SAR of novel tricyclic quinoxalinone inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1)
Miyashiro, J., Woods, K.W., Park, C.H., Liu, X., Shi, Y., Johnson, E.F., Bouska, J.J., Olson, A.M., Luo, Y., Fry, E.H., Giranda, V.L., Penning, T.D.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2009-03-09
Resolution2.300
CATH Insert Date11 Mar, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Mar, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3gjwA01 23 Mar, 2010 1.20.142.10 Assigned
3gjwA02 23 Mar, 2010 3.90.228.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P09874 PARP1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 1