PDB 3gjw
PDB Information
| PDB | 3GJW |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Synthesis and SAR of novel tricyclic quinoxalinone inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1)
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2009-03-09 |
| Resolution | 2.300 |
| CATH Insert Date | 11 Mar, 2010 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Mar, 2010 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3gjwA01 | 23 Mar, 2010 | 1.20.142.10 | Assigned |
| 3gjwA02 | 23 Mar, 2010 | 3.90.228.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
