PDB Information

PDB3GI3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and characterization of the N-phenyl-N'-naphthylurea class of p38 kinase inhibitors.
Cirillo, P.F., Hickey, E.R., Moss, N., Breitfelder, S., Betageri, R., Fadra, T., Gaenzler, F., Gilmore, T., Goldberg, D.R., Kamhi, V., Kirrane, T., Kroe, R.R., Madwed, J., Moriak, M., Netherton, M., Pargellis, C.A., Patel, U.R., Qian, K.C., Sharma, R., Sun, S., Swinamer, A., Torcellini, C., Takahashi, H., Tsang, M., Xiong, Z.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2009-03-05
Resolution2.400
CATH Insert Date01 Nov, 2009

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 01 Nov, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3gi3A01 26 Dec, 2009 3.30.200.20 Assigned
3gi3A02 26 Dec, 2009 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q16539 MK14_HUMAN Homo sapiens Mitogen-activated protein kinase 14