PDB 3g42
PDB Information
| PDB | 3G42 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Cricetulus griseus |
| Gene Source | Homo sapiens |
| Primary Citation | Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-alpha converting enzyme (TACE) inhibitors.
Bioorg.Med.Chem.
|
| Header | Hydrolase |
| Released | 2009-02-03 |
| Resolution | 2.100 |
| CATH Insert Date | 16 Aug, 2009 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Aug, 2009 | Chopped |
| B | 16 Aug, 2009 | Chopped |
| C | 16 Aug, 2009 | Chopped |
| D | 16 Aug, 2009 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3g42A00 | 13 Dec, 2009 | 3.40.390.10 | Assigned |
| 3g42B00 | 13 Dec, 2009 | 3.40.390.10 | Assigned |
| 3g42C00 | 13 Dec, 2009 | 3.40.390.10 | Assigned |
| 3g42D00 | 13 Dec, 2009 | 3.40.390.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P78536 | ADA17_HUMAN | Homo sapiens | Disintegrin and metalloproteinase domain-containing protein 17 |
| P78536 | ADA17_HUMAN | Homo sapiens | Disintegrin and metalloproteinase domain-containing protein 17 |
| P78536 | ADA17_HUMAN | Homo sapiens | Disintegrin and metalloproteinase domain-containing protein 17 |
| P78536 | ADA17_HUMAN | Homo sapiens | Disintegrin and metalloproteinase domain-containing protein 17 |
