PDB Information

PDB3G42
MethodX-RAY DIFFRACTION
Host OrganismCricetulus griseus
Gene SourceHomo sapiens
Primary Citation
Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-alpha converting enzyme (TACE) inhibitors.
Park, K., Gopalsamy, A., Aplasca, A., Ellingboe, J.W., Xu, W., Zhang, Y., Levin, J.I.
Bioorg.Med.Chem.
HeaderHydrolase
Released2009-02-03
Resolution2.100
CATH Insert Date16 Aug, 2009

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Chopped
C 16 Aug, 2009 Chopped
D 16 Aug, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3g42A00 13 Dec, 2009 3.40.390.10 Assigned
3g42B00 13 Dec, 2009 3.40.390.10 Assigned
3g42C00 13 Dec, 2009 3.40.390.10 Assigned
3g42D00 13 Dec, 2009 3.40.390.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17