PDB Information

PDB3FUG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Modulating retinoid X receptor with a series of (E)-3-[4-hydroxy-3-(3-alkoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)phenyl]acrylic acids and their 4-alkoxy isomers.
Perez Santin, E., Germain, P., Quillard, F., Khanwalkar, H., Rodriguez-Barrios, F., Gronemeyer, H., de Lera, A.R., Bourguet, W.
J.Med.Chem.
HeaderTranscription/Transcription Regulator
Released2009-01-14
Resolution2.000
CATH Insert Date16 Aug, 2009

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3fugA00 18 Mar, 2013 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P19793 RXRA_HUMAN Homo sapiens Retinoic acid receptor RXR-alpha
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2