PDB Information

PDB3FKT
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Discovery and X-ray Crystallographic Analysis of a Iminohydantoin Inhibitor of beta-Secretase
Barrow, J.C., Stauffer, S.R., Rittle, K.E., Ngo, P.L., Yang, M.S., Graham, S., McGaughey, G., Holloway, K., Tugusheva, S.K., Lai, M., Espeseth, A.S., Xu, M., Huang, Q., Zuck, P., Levorse, D.A., Hazuda, D., Vacca, J.P.
J.Med.Chem.
HeaderHydrolase
Released2008-12-17
Resolution1.900
CATH Insert Date22 Jan, 2009

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 Jan, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3fktA01 24 Jan, 2009 2.40.70.10 Assigned
3fktA02 24 Jan, 2009 2.40.70.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P56817 BACE1_HUMAN Homo sapiens Beta-secretase 1