PDB Information

PDB3F7G
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Orally bioavailable antagonists of inhibitor of apoptosis proteins based on an azabicyclooctane scaffold
Cohen, F., Alicke, B., Elliott, L.O., Flygare, J.A., Goncharov, T., Keteltas, S.F., Franklin, M.C., Frankovitz, S., Stephan, J.P., Tsui, V., Vucic, D., Wong, H., Fairbrother, W.J.
J.Med.Chem.
HeaderApoptosis
Released2008-11-09
Resolution2.300
CATH Insert Date19 Mar, 2009

PDB Images (11)

PDB Prints

PDB Chains (5)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Chopped
C 16 Aug, 2009 Chopped
D 16 Aug, 2009 Chopped
E 16 Aug, 2009 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
3f7gA00 04 Feb, 2013 1.10.1170.10 Assigned
3f7gB00 04 Feb, 2013 1.10.1170.10 Assigned
3f7gC00 04 Feb, 2013 1.10.1170.10 Assigned
3f7gD00 04 Feb, 2013 1.10.1170.10 Assigned
3f7gE00 04 Feb, 2013 1.10.1170.10 Assigned

UniProtKB Entries (5)

Accession Gene ID Taxon Description
Q96CA5 BIRC7_HUMAN Homo sapiens Baculoviral IAP repeat-containing protein 7
Q96CA5 BIRC7_HUMAN Homo sapiens Baculoviral IAP repeat-containing protein 7
Q96CA5 BIRC7_HUMAN Homo sapiens Baculoviral IAP repeat-containing protein 7
Q96CA5 BIRC7_HUMAN Homo sapiens Baculoviral IAP repeat-containing protein 7
Q96CA5 BIRC7_HUMAN Homo sapiens Baculoviral IAP repeat-containing protein 7