PDB Information

PDB3F3V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceGallus gallus
Primary Citation
Hybrid compound design to overcome the gatekeeper T338M mutation in cSrc
Getlik, M., Grutter, C., Simard, J.R., Kluter, S., Rabiller, M., Rode, H.B., Robubi, A., Rauh, D.
J.Med.Chem.
HeaderTransferase
Released2008-10-31
Resolution2.600
CATH Insert Date16 Aug, 2009

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2009 Chopped
B 16 Aug, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3f3vA01 07 Oct, 2009 3.30.200.20 Assigned
3f3vA02 07 Oct, 2009 1.10.510.10 Assigned
3f3vB01 07 Oct, 2009 3.30.200.20 Assigned
3f3vB02 07 Oct, 2009 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00523 SRC_CHICK Gallus gallus Proto-oncogene tyrosine-protein kinase Src
P00523 SRC_CHICK Gallus gallus Proto-oncogene tyrosine-protein kinase Src