PDB 3eqr

PDB Links
Overview

PDB Information

PDB	3EQR
Method	X-RAY DIFFRACTION
Host Organism	Insect cells
Gene Source	Homo sapiens
Primary Citation	Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors. Kopecky, D.J., Hao, X., Chen, Y., Fu, J., Jiao, X., Jaen, J.C., Cardozo, M.G., Liu, J., Wang, Z., Walker, N.P., Wesche, H., Li, S., Farrelly, E., Xiao, S.H., Kayser, F. Bioorg.Med.Chem.Lett.
Header	Transferase
Released	2008-10-01
Resolution	2.000
CATH Insert Date	07 Dec, 2008

PDB Images (7)

Image of CATH 3eqr

3eqr

PDB 3eqr

Image of CATH 3eqrA

3eqrA

PDB Chain 3eqrA

Image of CATH 3eqrB

3eqrB

PDB Chain 3eqrB

Image of CATH 3eqrA01

3eqrA01

CATH Domain 3eqrA01

Image of CATH 3eqrA02

3eqrA02

CATH Domain 3eqrA02

Image of CATH 3eqrB01

3eqrB01

CATH Domain 3eqrB01

Image of CATH 3eqrB02

3eqrB02

CATH Domain 3eqrB02

PDB Prints

PDB Chains (2)

Chain ID	Date inserted into CATH	CATH Status
A	07 Dec, 2008	Chopped
B	07 Dec, 2008	Chopped

CATH Domains (4)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
3eqrA01	31 Mar, 2009	3.30.200.20	Assigned
3eqrA02	31 Mar, 2009	1.10.510.10	Assigned
3eqrB01	31 Mar, 2009	3.30.200.20	Assigned
3eqrB02	31 Mar, 2009	1.10.510.10	Assigned

UniProtKB Entries (2)

Accession	Gene ID	Taxon	Description
Q07912	ACK1_HUMAN	Homo sapiens	Activated CDC42 kinase 1
Q07912	ACK1_HUMAN	Homo sapiens	Activated CDC42 kinase 1