PDB Information

PDB3EQP
MethodX-RAY DIFFRACTION
Host OrganismInsect cells
Gene SourceHomo sapiens
Primary Citation
Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors.
Kopecky, D.J., Hao, X., Chen, Y., Fu, J., Jiao, X., Jaen, J.C., Cardozo, M.G., Liu, J., Wang, Z., Walker, N.P., Wesche, H., Li, S., Farrelly, E., Xiao, S.H., Kayser, F.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-10-01
Resolution2.300
CATH Insert Date07 Dec, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Dec, 2008 Chopped
B 07 Dec, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3eqpA01 31 Mar, 2009 3.30.200.20 Assigned
3eqpA02 31 Mar, 2009 1.10.510.10 Assigned
3eqpB01 31 Mar, 2009 3.30.200.20 Assigned
3eqpB02 31 Mar, 2009 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q07912 ACK1_HUMAN Homo sapiens Activated CDC42 kinase 1
Q07912 ACK1_HUMAN Homo sapiens Activated CDC42 kinase 1