PDB Information

PDB3ENS
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Design, Structure-Activity Relationships, X-ray Crystal Structure, and Energetic Contributions of a Critical P1 Pharmacophore: 3-Chloroindole-7-yl-Based Factor Xa Inhibitors.
Shi, Y., Sitkoff, D., Zhang, J., Klei, H.E., Kish, K., Liu, E.C., Hartl, K.S., Seiler, S.M., Chang, M., Huang, C., Youssef, S., Steinbacher, T.E., Schumacher, W.A., Grazier, N., Pudzianowski, A., Apedo, A., Discenza, L., Yanchunas, J., Stein, P.D., Atwal, K.S.
J.Med.Chem.
HeaderHydrolase, Blood Clotting
Released2008-09-25
Resolution2.300
CATH Insert Date01 Jan, 2009

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 01 Jan, 2009 Chopped
B 01 Jan, 2009 Chopped
C 01 Jan, 2009 Chopped
D 01 Jan, 2009 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3ensA01 07 Jan, 2009 2.10.25.10 Assigned
3ensA02 07 Jan, 2009 2.10.25.10 Assigned
3ensB01 07 Jan, 2009 2.40.10.10 Assigned
3ensB02 07 Jan, 2009 2.40.10.10 Assigned
3ensC01 07 Jan, 2009 2.10.25.10 Assigned
3ensC02 07 Jan, 2009 2.10.25.10 Assigned
3ensD01 07 Jan, 2009 2.40.10.10 Assigned
3ensD02 07 Jan, 2009 2.40.10.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X