PDB Information

PDB3EJ1
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Synthesis and evaluation of pyrazolo[1,5-b]pyridazines as selective cyclin dependent kinase inhibitors.
Stevens, K.L., Reno, M.J., Alberti, J.B., Price, D.J., Kane-Carson, L.S., Knick, V.B., Shewchuk, L.M., Hassell, A.M., Veal, J.M., Davis, S.T., Griffin, R.J., Peel, M.R.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Cell Cycle
Released2008-09-17
Resolution3.220
CATH Insert Date23 Oct, 2008

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 23 Oct, 2008 Chopped
B 23 Oct, 2008 Chopped
C 23 Oct, 2008 Chopped
D 23 Oct, 2008 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3ej1A01 25 Oct, 2008 3.30.200.20 Assigned
3ej1A02 25 Oct, 2008 1.10.510.10 Assigned
3ej1B01 25 Oct, 2008 1.10.472.10 Assigned
3ej1B02 25 Oct, 2008 1.10.472.10 Assigned
3ej1C01 25 Oct, 2008 3.30.200.20 Assigned
3ej1C02 25 Oct, 2008 1.10.510.10 Assigned
3ej1D01 25 Oct, 2008 1.10.472.10 Assigned
3ej1D02 25 Oct, 2008 1.10.472.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2