PDB Information

PDB3E8E
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceBos taurus
Primary Citation
Aminofurazans as potent inhibitors of AKT kinase
Rouse, M.B., Seefeld, M.A., Leber, J.D., McNulty, K.C., Sun, L., Miller, W.H., Zhang, S., Minthorn, E.A., Concha, N.O., Choudhry, A.E., Schaber, M.D., Heerding, D.A.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-08-19
Resolution2.000
CATH Insert Date20 Nov, 2008

PDB Images (25)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 20 Nov, 2008 Chopped
B 20 Nov, 2008 Chopped
C 20 Nov, 2008 Rejected
E 20 Nov, 2008 Chopped
F 20 Nov, 2008 Rejected
G 20 Nov, 2008 Rejected
I 20 Nov, 2008 Chopped
J 20 Nov, 2008 Rejected
L 20 Nov, 2008 Chopped
N 20 Nov, 2008 Rejected
P 20 Nov, 2008 Chopped
Q 20 Nov, 2008 Rejected

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
3e8eA01 08 Dec, 2008 1.10.510.10 Assigned
3e8eA02 08 Dec, 2008 3.30.200.20 Assigned
3e8eB01 08 Dec, 2008 1.10.510.10 Assigned
3e8eB02 08 Dec, 2008 3.30.200.20 Assigned
3e8eE01 08 Dec, 2008 1.10.510.10 Assigned
3e8eE02 08 Dec, 2008 3.30.200.20 Assigned
3e8eI01 08 Dec, 2008 1.10.510.10 Assigned
3e8eI02 08 Dec, 2008 3.30.200.20 Assigned
3e8eL01 08 Dec, 2008 1.10.510.10 Assigned
3e8eL02 08 Dec, 2008 3.30.200.20 Assigned
3e8eP01 08 Dec, 2008 1.10.510.10 Assigned
3e8eP02 08 Dec, 2008 3.30.200.20 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha