PDB Information

PDB3E63
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Fragment-based discovery of JAK-2 inhibitors.
Antonysamy, S., Hirst, G., Park, F., Sprengeler, P., Stappenbeck, F., Steensma, R., Wilson, M., Wong, M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-08-14
Resolution1.900
CATH Insert Date16 Oct, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Oct, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3e63A01 17 Oct, 2008 3.30.200.20 Assigned
3e63A02 17 Oct, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2