PDB Information

PDB3D4Q
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Potent and selective pyrazole-based inhibitors of B-Raf kinase.
Hansen, J.D., Grina, J., Newhouse, B., Welch, M., Topalov, G., Littman, N., Callejo, M., Gloor, S., Martinson, M., Laird, E., Brandhuber, B.J., Vigers, G., Morales, T., Woessner, R., Randolph, N., Lyssikatos, J., Olivero, A.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-05-14
Resolution2.800
CATH Insert Date24 Aug, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 24 Aug, 2008 Chopped
B 24 Aug, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3d4qA01 25 Aug, 2008 3.30.200.20 Assigned
3d4qA02 25 Aug, 2008 1.10.510.10 Assigned
3d4qB01 25 Aug, 2008 3.30.200.20 Assigned
3d4qB02 25 Aug, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf